Peptide Active Data Details
Basic Peptide Information
DICL ID
DICL_Pep_04380
Ion Channel
Sodium channel type 5 subunit alpha
Peptide Function
Inhibitor
Gene Name
Scn5a
Activity Data (nM)
IC50
72 nM
Ki
Not available
EC50
Not available
Kd
Not available
Biologically Active
Not specified
Sequence Information
Peptide Sequence
DCLGFLWKCNPSNDKCCRPNLVCSRKDKWCKYQI
Peptide UniProt Accession
UniParc
Not available
Peptide Synonyms/Alias
Paurtx3; recombinant Paurtx-3 (rPaurtx-3)
Peptide Species
Paraphysa scrofa (Chilean copper tarantula) (Phrixotrichus auratus)
Peptide Name
Beta-theraphotoxin-Ps1a
CAS Number
Not available
Experimental Conditions
pH
pH 7.4
Holding Potential (mV)
−90 mV
Temperature
22–25 °C
Test Method
Patch-clamping
Test Species
HEK293T cell (Homo sapiens embryonic kidney 293T cell)
Binding Information
Binding Site
Not specified
Binding Site Residue
Not specified
Ion Channel Information
Gene Abbreviation (ABB)
VGSCs
Ion Channel UniProt Accession
Source Organism
Rattus norvegicus (Rat)
References & Disease Information
Disease
Not specified
PubChem CID
Not available
URL
Not available
PMID
Patent
Not available